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Amy M. Kucken, Jeremy A. Teissére, James Seffinga-Clark, David A. Wagner, Cynthia Czajkowski. Structural Requirements for Imidazobenzodiazepine Binding to GABA A Receptors. Molecular Pharmacology 2003 , 63 (2) , 289-296. 63 (2) , 289-296. https://doi.org/10.1124/mol.63.2.289

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Eduardo Cortés Cortés, Isidro Ebromares Martínez, Olivia García Mellado. Synthesis and spectral properties of 7-chloro-5-[( o - and p -R 1 )phenyl]-1-R 2 -3 H -[1,4]benzodiazepin-2-ones. Journal of Heterocyclic Chemistry 2002 , 39 (6) , 1189-1193. 39 (6) , 1189-1193. https://doi.org/10.1002/jhet.5570390612

M.Teresa Herrero, Imanol Tellitu, Esther Domı́nguez, Isabel Moreno, Raúl SanMartı́n. A novel and efficient iodine(III)-mediated access to 1,4-benzodiazepin-2-ones. Tetrahedron Letters 2002 , 43 (46) , 8273-8275. 43 (46) , 8273-8275. https://doi.org/10.1016/S0040-4039(02)02019-1

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Takashi Miki, Masakuni Kori, Akira Fujishima, Hiroshi Mabuchi, Ryu-ichi Tozawa, Masahira Nakamura, Yasuo Sugiyama, Hidefumi Yukimasa. Syntheses of fused heterocyclic compounds and their inhibitory activities for squalene synthase. Bioorganic & Medicinal Chemistry 2002 , 10 (2) , 385-400. 10 (2) , 385-400. https://doi.org/10.1016/S0968-0896(01)00289-9

Lalit Kumar Baregama, Bhawani Singh, G.L. Talesara. SYNTHESIS OF 3-ALKOXY-(SUBSTITUTED ARYL) BIGUANIDINO-4-METHYL-2,3-DIHYDRO(1H)-1,5-BENZODIAZEPINE-2-ONES AND RELATED COMPOUNDS. Heterocyclic Communications 2002 , 8 (6) 8 (6) https://doi.org/10.1515/HC.2002.8.6.607

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Eduardo Cortés Cortés, Raúl Salazar Franco, Olivia García Mellado. Synthesis and spectral properties of 2-[(o- and p-substituted)aminophenyl] -3 H -5-[(o- and p -substituted)phenyl]-7-chloro-1,4-benzodiazepines. Journal of Heterocyclic Chemistry 2001 , 38 (3) , 663-669. 38 (3) , 663-669. https://doi.org/10.1002/jhet.5570380320

Qi-Han Zhang, Jia-Xi Xu. A Novel Conversion of 2, 4-Diaryl-2, 3-dihydro-1 H-1, 5-benzodiazepines into 2, 4-Diaryl-3 H-1, 5-benzodiazepines. Chinese Journal of Chemistry 2001 , 19 (4) , 378-380. 19 (4) , 378-380. https://doi.org/10.1002/cjoc.20010190411

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Jatinder P. Bassin, Martin J. Frearson, Karim Al-nawwar. Synthesis of Benzo[d]Benzo[2,3][1,4]Diazepino[1,7- b ]Isothiazole, a New Heterocyclic Ring System. Synthetic Communications 2000 , 30 (16) , 2961-2965. 30 (16) , 2961-2965. https://doi.org/10.1080/00397910008087446

Helmut Quast, Svetlana Ivanova, Eva-Maria Peters, Karl Peters. Ring Expansion of 2-Alkylidenedihydroquinazolines to Iminodihydro-1,4-benzodiazepines by Methanesulfonyl and Trifluoromethanesulfonyl Azide. European Journal of Organic Chemistry 2000 , 2000 (8) , 1577-1587. 2000 (8) , 1577-1587. https://doi.org/10.1002/(SICI)1099-0690(200004)2000:8<1577::AID-EJOC1577>3.0.CO;2-6

Benjamin E Blass, Thomas M Burt, Song Liu, David E Portlock, Erin M Swing. A facile KF/Al2O3 mediated, selective alkylation of benzodiazepin-2,5-diones. Tetrahedron Letters 2000 , 41 (13) , 2063-2066. 41 (13) , 2063-2066. https://doi.org/10.1016/S0040-4039(00)00115-5

Helmut Quast, Svetlana Ivanova, Eva-Maria Peters, Karl Peters. Ring Expansion of 2-Alkylidenedihydroquinolines to 2-Iminodihydro-1-benzazepines by Phenyl, Methanesulphonyl, and Trifluoromethanesulphonyl Azide[1]. European Journal of Organic Chemistry 2000 , 2000 (3) , 507-520. 2000 (3) , 507-520. https://doi.org/10.1002/(SICI)1099-0690(200002)2000:3<507::AID-EJOC507>3.0.CO;2-V

Jiaxi Xu, Liangbi Chen. Synthesis of oxazirino[2,3-a][1,5]benzodiazepines by oxidation of 1H-1,5-benzodiazepines withm-chloroperbenzoic acid (MCPBA). Heteroatom Chemistry 2000 , 11 (2) , 158-162. 11 (2) , 158-162. https://doi.org/10.1002/(SICI)1098-1071(2000)11:2<158::AID-HC12>3.0.CO;2-G

Achim Escherich, J�rgen Lutz, Chantal Escrieut, Daniel Fourmy, A. Stephanie van Neuren, Gerhard M�ller, Andrea Schafferhans, Gerhard Klebe, Luis Moroder. Peptide/benzodiazepine hybrids as ligands of CCKA and CCKB receptors. Biopolymers 2000 , 56 (2) , 55-76. 56 (2) , 55-76. https://doi.org/10.1002/1097-0282(2000)56:2<55::AID-BIP1052>3.0.CO;2-M

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Katja Heinig, Jack Henion. Fast liquid chromatographic–mass spectrometric determination of pharmaceutical compounds. Journal of Chromatography B: Biomedical Sciences and Applications 1999 , 732 (2) , 445-458. 732 (2) , 445-458. https://doi.org/10.1016/S0378-4347(99)00313-8

Jiaxi Xu, Bo Liang, Sheng Jin. SYNTHESIS OF 1,5-BENZOTHIAZEPINE-1-OXIDE/-1,1-DIOXIDE DERIVATIVES AND 1,2-OXAZIRINO[2,3- a ] [1,5] BENZODIAZEPINE. Phosphorus, Sulfur, and Silicon and the Related Elements 1999 , 152 (1) , 1-8. 152 (1) , 1-8. https://doi.org/10.1080/10426509908031612

Latha Ramdas, Barry A. Bunnin, Matthew J. Plunkett, Gongqin Sun, Jonathan Ellman, Gary Gallick, Raymond J.A. Budde. Benzodiazepine Compounds as Inhibitors of the Src Protein Tyrosine Kinase: Screening of a Combinatorial Library of 1,4-Benzodiazepines. Archives of Biochemistry and Biophysics 1999 , 368 (2) , 394-400. 368 (2) , 394-400. https://doi.org/10.1006/abbi.1999.1313

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Eduardo Cortés Cortés, Maria Paz Sánchez Bravo. Synthesis and spectral properties of 2,3-dihydro-2-[( o - and p -substituted)anilinylidene]-1 H -4-( p -methylphenyl)-7-[( o - and p -methyl)phenoxy]-1,5-benzodiazepines. Journal of Heterocyclic Chemistry 1999 , 36 (3) , 611-615. 36 (3) , 611-615. https://doi.org/10.1002/jhet.5570360306

Xavier Doisy, Mouloud Dekhane, Mireille Le Hyaric, Jean-François Rousseau, Sunil K Singh, Suan Tan, Valérie Guilleminot, Hans Schoemaker, Mireille Sevrin, Pascal George, Pierre Potier, Robert H Dodd. Synthesis and benzodiazepine receptor (ω receptor) affinities of 3-substituted derivatives of pyrrolo[2,3-c]pyridine-5-carboxylate, a novel class of ω1 selective ligands1This article is dedicated to the memory of our friend and colleague, Sir Derek Barton.1. Bioorganic & Medicinal Chemistry 1999 , 7 (5) , 921-932. 7 (5) , 921-932. https://doi.org/10.1016/S0968-0896(99)00053-X

Charles Y. Fiakpui, Oludotun A. Phillips, K. S. Keshava Murthy, Edward E. Knaus. Synthesis and anticonvulsant activities of 5-(2-Chlorophenyl)-7 H -pyrido[4,3- f ][1,2,4]triazolo[4,3- a ][1,4]diazepines. Journal of Heterocyclic Chemistry 1999 , 36 (2) , 377-380. 36 (2) , 377-380. https://doi.org/10.1002/jhet.5570360208

K.S. Keshava Murthy, Edward E. Knaus. Synthesis of pyrimido[1,4]diazepin-2-one analogs and their evaluation as anticonvulsant agents. Drug Development Research 1999 , 46 (2) , 155-162. 46 (2) , 155-162. https://doi.org/10.1002/(SICI)1098-2299(199902)46:2<155::AID-DDR9>3.0.CO;2-W

Jiaxi Xu, Sheng Jin. Thermal cycloaddition reaction of symmetrical and unsymmetrical ?-diazo-?-diketones with 4-aryl-2-methyl-2,3-dihydro-1,5-benzothia/diazepines. Heteroatom Chemistry 1999 , 10 (1) , 35-40. 10 (1) , 35-40. https://doi.org/10.1002/(SICI)1098-1071(1999)10:1<35::AID-HC7>3.0.CO;2-#

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Giovanni Minghetti, Antonio Zucca, Maria Agostina Cinellu, Sergio Stoccoro, Mario Manassero*, Mirella Sansoni. C(3) aurated 1,4-benzodiazepin-2-ones. Synthesis and characterization. Crystal structure of (L)Au[P(C6H4CH3-4)3] (HL=7-chloro-1,3-dihydro-1-methyl-5-phenyl-2H-1,4-benzodiazepin-2-one, DIAZEPAM). Journal of Organometallic Chemistry 1998 , 553 (1-2) , 405-415. 553 (1-2) , 405-415. https://doi.org/10.1016/S0022-328X(97)00624-4

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